erno Laslo

Transcrição

erno Laslo
Title (en)
Nitrocatechol derivates as COMT inhibitors administered with a specific dosage regime
Title (de)
Catechol Derivate als COMT-Hemmer eingenommen mit einer spezifischen Dosierungsanleitung
Title (fr)
Dérivés du catéchol comme inhibiteurs de la COMT administrés avec une posologie spécifique
Publication
EP 2481410 B1 20160713 (EN)
Application
EP 12163797 A 20071010
Priority
• EP 07834911 A 20071010
• EP 07002091 A 20070131
• EP 12163797 A 20071010
Abstract (en)
[origin: WO2008094053A1] The invention relates to the use of an oxodiazolyl compound (I) for the preparation of a medicament for the prevention or
treatment of central and peripheral nervous system associated disorders, wherein said medicament is administered according to a dosing regimen
having a dosing periodicity ranging from about twice a day to about once every other day.
Inventor
• LEARMONTH DAVID ALEXANDER (PT)
• KISS LASZLO ERNO (PT)
• LEAL PALMA PEDRO NUNO (PT)
• DOS SANTOS FERREIRA HUMBERTO (PT)
• VIEIRA ARAÚJO SOARES DA SILVA PATRÍCIO MANUEL (PT)
Applicant
BIAL PORTELA & CA SA (PT)
IPC 8 full level (invention and additional information)
A61K 31/4439 (2006.01); A61P 25/16 (2006.01)
CPC (invention and additional information)
C07D 413/04 (2013.01); A61K 9/20 (2013.01); A61K 31/198 (2013.01); A61K 31/4439 (2013.01); A61K 45/06 (2013.01)
Citation (examination)
None
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR
Designated extension state (EPC)
HR
EPO simple patent family
WO 2008094053 A1 20080807; AR 065098 A1 20090513; AU 2007346018 A1 20080807; AU 2007346018 A2 20110421; BR PI0721213 A2
20140318; CA 2678391 A1 20080807; CN 101631548 A 20100120; CN 101631548 B 20140827; EP 2124947 A1 20091202; EP 2481410 A1
20120801; EP 2481410 B1 20160713; IL 200020 D0 20100415; JP 2011500506 A 20110106; JP 5517629 B2 20140611; KR 101522157 B1
20150528; KR 20090104859 A 20091006; MX 2009008051 A 20090812; NO 20092905 A 20091029; RU 2009132188 A 20110310; RU 2518483
C2 20140610; US 2010113529 A1 20100506; US 2013331416 A1 20131212; US 2016009699 A1 20160114; US 8524746 B2 20130903; ZA
200905940 B 20100526
INPADOC legal status
2016-08-25 [REG DE R096] DPMA PUBLICATION OF MENTIONED EP PATENT GRANT
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2016-07-15 [REG AT REF] REFERENCE TO AT NUMBER (EP PATENT ENTERS AUSTRIAN NATIONAL PHASE)
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- Country of Ref Document : AT
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2016-07-15 [REG CH EP] ENTRY IN THE NATIONAL PHASE
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2016-07-13 [AC] DIVISIONAL APPLICATION (ART. 76) OF:
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- Kind Code of Ref Document : B1
- Designated State(s) : AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI
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2016-07-13 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO
- Countries concerned : HR
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2016-07-13 [REG GB FG4D] EUROPEAN PATENT GRANTED
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2016-01-20 [INTG] ANNOUNCEMENT OF INTENTION TO GRANT
- Effective date : 20151221
2016-01-20 [RIN1] INVENTOR (CORRECTION)
- Inventor name : DOS SANTOS FERREIRA, HUMBERTO
2016-01-20 [RIN1] INVENTOR (CORRECTION)
- Inventor name : KISS, LASZLO ERNO
2016-01-20 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LEAL PALMA, PEDRO NUNO
2016-01-20 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LEARMONTH, DAVID ALEXANDER
2016-01-20 [RIN1] INVENTOR (CORRECTION)
- Inventor name : VIEIRA ARAUJO SOARES DA SILVA, PATRICIO MANUEL
2015-11-04 [RIN1] INVENTOR (CORRECTION)
- Inventor name : DOS SANTOS FERREIRA, HUMBERTO
2015-11-04 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LASZLO, ERNO KISS
2015-11-04 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LEAL PALMA, PEDRO NUNO
2015-11-04 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LEARMONTH, DAVID ALEXANDER
2015-11-04 [RIN1] INVENTOR (CORRECTION)
- Inventor name : VIEIRA ARAUJO SOARES DA SILVA, PATRICIO MANUEL
2013-05-15 [17Q] FIRST EXAMINATION REPORT
- Effective date : 20130415
2013-03-06 [17P] REQUEST FOR EXAMINATION FILED
- Effective date : 20130125
2012-09-05 [RIN1] INVENTOR (CORRECTION)
- Inventor name : ARAUJO SOARES DA SILVA, PATRICIO MANUEL VIEIRA
2012-09-05 [RIN1] INVENTOR (CORRECTION)
- Inventor name : DOS SANTOS FERREIRA, HUMBERTO
2012-09-05 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LASZLO, ERNO KISS
2012-09-05 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LEAL PALMA, PEDRO NUNO
2012-09-05 [RIN1] INVENTOR (CORRECTION)
- Inventor name : LEARMONTH, DAVID ALEXANDER
2012-08-01 [AC] DIVISIONAL APPLICATION (ART. 76) OF:
- Ref Document Number : 2124947
- Country of Ref Document : EP
- Kind Code of Ref Document : P
2012-08-01 [AK] DESIGNATED CONTRACTING STATES:
- Kind Code of Ref Document : A1
- Designated State(s) : AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI
SK TR
2012-08-01 [AX] REQUEST FOR EXTENSION OF THE EUROPEAN PATENT TO
- Countries concerned : HR

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